- Endothelin receptor antagonist
A endothelin receptor antagonist (ERA) is a drug which blocks
Two main kinds of ERAs exist:
* selective ERA (e.g.
sitaxsentan), which affect endothelin A.
* dual ERAs,(e.g.
bosentan) which affect both endothelin A and B . [ [http://cvpharmacology.com/vasodilator/ETblockers.htm Endothelin receptor antagonists ] ]
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